发明名称 IMIDIAZOLE DERIVATIVES AND THEIR USE AS AGONISTS SELECTIVE AT ALPHA 2B OR 2B/2C ADRENERGIC RECEPTORS
摘要 Methods and compounds for the treatment of conditions including pain, particularly chronic pain, glaucoma or elevated intraocular pressure with reduced cardiovascular or sedative side effects. Also included are methods of making and using such compounds.
申请公布号 EP1370533(A2) 申请公布日期 2003.12.17
申请号 EP20020723489 申请日期 2002.03.13
申请人 ALLERGAN, INC. 发明人 CHOW, KEN;GIL, DANIEL, W.;BURKE, JAMES, A.;HARCOURT, DALE, A.;GARST, MICHAEL, E.;WHEELER, LARRY, A.;MUNK, STEPHEN, A.;GOMEZ, DARIO, G.
分类号 C07D233/58;A61K31/4164;A61K31/4178;A61K31/421;A61K31/435;A61K31/4709;A61K31/4725;A61K31/498;A61K31/538;A61P1/12;A61P7/12;A61P9/00;A61P9/04;A61P9/10;A61P9/12;A61P25/02;A61P25/04;A61P25/14;A61P25/18;A61P25/22;A61P25/24;A61P25/28;A61P27/02;A61P27/06;A61P27/16;A61P43/00;C07D233/06;C07D233/10;C07D233/54;C07D233/64;C07D233/84;C07D263/28;C07D401/06;C07D403/06;C07D405/06;C07D409/06;C07D413/12;C07D495/04;(IPC1-7):C07D233/54;A61K31/416 主分类号 C07D233/58
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