发明名称 |
N-SUBSTITUTED NON-ARYL HETEROCYCLIC ANTAGONISTS NMDA/NR2B |
摘要 |
Compounds represented by Formula (I): (I)or pharmaceutically acceptable salts thereof, are effective as NMDA NR2B antagonists useful for relieving pain. (I)
|
申请公布号 |
UA75392(C2) |
申请公布日期 |
2003.12.15 |
申请号 |
UA20030098659 |
申请日期 |
2002.02.20 |
申请人 |
MERCK & CO., INC. |
发明人 |
KLAYBORN CRISTOPHER F.;BUTCHER JOHN U.;CLAIRMON DAVID A.;LIBBI BRAYAN E.;LIVERTON NIGEL G.;MANSON PETER M.;NGUYEN KEVIN T.;MCCOLI JOHN A. |
分类号 |
A61K31/454;A61K31/444;A61K31/4709;A61K31/4745;A61K31/497;A61K31/501;A61K31/506;A61K31/517;A61K31/519;A61K31/52;A61K31/525;A61P25/04;A61P25/06;A61P25/16;A61P25/18;A61P25/22;A61P25/24;A61P25/28;A61P29/02;C07D401/12;C07D403/12;C07D409/14;C07D413/12;C07D417/12;C07D451/02;C07D471/04;C07D471/08;C07D473/16;C07D473/34;C07D475/00;C07D475/06;C07D475/08;C07D487/04;C07D519/00 |
主分类号 |
A61K31/454 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|