发明名称 NOVEL CONAZOLE CRYSTALLINE FORMS AND RELATED PROCESSES, PHARMACEUTICAL COMPOSITIONS AND METHODS
摘要 The invention provides novel soluble conazole crystalline forms (e.g.itraconazole, posaconazole and saperconazole) that includes salts, co-crystals and related solvates useful as pharmaceuticals. The invention also provides pharmaceutical compositions comprising, and processes for making, these conazole crystalline forms. Methods of using such compositions for the treatment or prevention of systemic and local fungal, yeast, and dermatophyte infections are also provided.
申请公布号 WO03101392(A2) 申请公布日期 2003.12.11
申请号 WO2003US17184 申请日期 2003.05.30
申请人 TRANSFORM PHARMACEUTICALS, INC.;REMENAR, JULIUS;MACPHEE, MICHAEL;PETERSON, MATTHEW, LYNN;MORISSETTE, SHERRY, L.;ALMARSSON, OM 发明人 REMENAR, JULIUS;MACPHEE, MICHAEL;PETERSON, MATTHEW, LYNN;MORISSETTE, SHERRY, L.;ALMARSSON, OM
分类号 A61K9/00;A61K9/16;A61K9/64;A61K31/496;A61K47/10;A61K47/32;A61P17/00;A61P25/00;A61P31/04;A61P31/10;B01D9/02;C07C57/15;C07C59/255;C07C309/29;C07D233/74;C07D405/14;G01N33/15 主分类号 A61K9/00
代理机构 代理人
主权项
地址