发明名称 |
PHENYL-THIOPHENE TYPE VITAMIN D RECEPTOR MODULATORS |
摘要 |
The present invention relates to novel, non-secosteroidal, phenyl-thiophene compounds with vitamin D receptor (VDR) modulating activity that are less hypercalcemic than 1.alpha.,25 dihydroxy vitamin D3. These compounds are useful for treating bone disease and psoriasis.
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申请公布号 |
CA2485503(A1) |
申请公布日期 |
2003.12.11 |
申请号 |
CA20032485503 |
申请日期 |
2003.05.22 |
申请人 |
ELI LILY AND COMPANY |
发明人 |
JONES, CHARLES DAVID;GAJEWSKI, ROBERT PETER;LINEBARGER, JARED HARRIS;LU, JIANLIANG;MA, TIANWEI;SIMARD, TODD PARKER;STITES, RYAN EDWARD;BUNEL, EMILIO ENRIQUE;DAHNKE, KARL ROBERT;YEE, YING KWONG;NAGPAL, SUNIL |
分类号 |
C07D333/16;A61K31/381;A61K31/4025;A61K31/41;A61K31/505;A61P3/02;A61P3/10;A61P13/12;A61P17/02;A61P17/06;A61P17/10;A61P17/14;A61P19/00;A61P19/02;A61P19/10;A61P25/28;A61P29/00;A61P35/00;A61P43/00;C07D333/18;C07D333/20;C07D333/22;C07D333/24;C07D333/34;C07D333/38;C07D333/40;C07D409/06;C07D409/12;C07D413/04;C07F9/6553;(IPC1-7):C07D333/38;C07D409/04;A61K31/401;A61K31/424 |
主分类号 |
C07D333/16 |
代理机构 |
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代理人 |
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地址 |
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