发明名称 PHENYL-THIOPHENE TYPE VITAMIN D RECEPTOR MODULATORS
摘要 The present invention relates to novel, non-secosteroidal, phenyl-thiophene compounds with vitamin D receptor (VDR) modulating activity that are less hypercalcemic than 1.alpha.,25 dihydroxy vitamin D3. These compounds are useful for treating bone disease and psoriasis.
申请公布号 CA2485503(A1) 申请公布日期 2003.12.11
申请号 CA20032485503 申请日期 2003.05.22
申请人 ELI LILY AND COMPANY 发明人 JONES, CHARLES DAVID;GAJEWSKI, ROBERT PETER;LINEBARGER, JARED HARRIS;LU, JIANLIANG;MA, TIANWEI;SIMARD, TODD PARKER;STITES, RYAN EDWARD;BUNEL, EMILIO ENRIQUE;DAHNKE, KARL ROBERT;YEE, YING KWONG;NAGPAL, SUNIL
分类号 C07D333/16;A61K31/381;A61K31/4025;A61K31/41;A61K31/505;A61P3/02;A61P3/10;A61P13/12;A61P17/02;A61P17/06;A61P17/10;A61P17/14;A61P19/00;A61P19/02;A61P19/10;A61P25/28;A61P29/00;A61P35/00;A61P43/00;C07D333/18;C07D333/20;C07D333/22;C07D333/24;C07D333/34;C07D333/38;C07D333/40;C07D409/06;C07D409/12;C07D413/04;C07F9/6553;(IPC1-7):C07D333/38;C07D409/04;A61K31/401;A61K31/424 主分类号 C07D333/16
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