发明名称 HIV protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis
摘要 Compounds of the formula: where the formula variables are as defined herein, are disclosed that advantageously inhibit or block the biological activity of the HIV protease. These compounds, as well as pharmaceutical compositions containing these compounds, are useful for treating patients or hosts infected with the HIV virus. Intermediates and synthetic methods for preparing such compounds are also described.
申请公布号 US2003225071(A1) 申请公布日期 2003.12.04
申请号 US20020166979 申请日期 2002.06.11
申请人 CANAN KOCH STACIE S.;ALEXANDER THERESE N.;BARVIAN MARK;BOLTON GARY;BOYER FREDRICK E.;BURKE BENJAMIN J.;HOLLER TOD;JEWELL TANYA M.;JOSYULA VARA PRASAD;KUCERA DAVID J.;LINTON MARIA A.;MACHAK JEFFREY J.;MITCHELL LENNERT J.;MURPHY SEAN T.;REICH SIEGFRIED H.;SKALITZKY DONALD J.;TATLOCK JOHN H.;VARNEY MICHAEL D.;VIRGIL SCOTT C.;WEBBER STEPHEN E.;WORLAND STEPHEN T.;MELNICK MICHAEL 发明人 CANAN KOCH STACIE S.;ALEXANDER THERESE N.;BARVIAN MARK;BOLTON GARY;BOYER FREDRICK E.;BURKE BENJAMIN J.;HOLLER TOD;JEWELL TANYA M.;JOSYULA VARA PRASAD;KUCERA DAVID J.;LINTON MARIA A.;MACHAK JEFFREY J.;MITCHELL LENNERT J.;MURPHY SEAN T.;REICH SIEGFRIED H.;SKALITZKY DONALD J.;TATLOCK JOHN H.;VARNEY MICHAEL D.;VIRGIL SCOTT C.;WEBBER STEPHEN E.;WORLAND STEPHEN T.;MELNICK MICHAEL
分类号 C07D277/04;A61K31/40;A61K31/401;A61K31/4025;A61K31/421;A61K31/422;A61K31/425;A61K31/426;A61K31/427;A61K31/428;A61K31/435;A61K31/439;A61K31/4439;A61K31/454;A61K31/4709;A61K31/472;A61K31/501;A61K31/5377;A61K31/541;A61K38/04;A61K45/00;A61P31/00;A61P31/12;A61P31/18;A61P37/02;A61P43/00;C07D207/09;C07D207/16;C07D207/24;C07D209/52;C07D213/38;C07D217/26;C07D231/12;C07D263/04;C07D263/06;C07D277/00;C07D277/06;C07D277/20;C07D277/28;C07D277/32;C07D277/38;C07D277/60;C07D295/13;C07D307/52;C07D403/12;C07D405/12;C07D409/12;C07D413/12;C07D417/12;C07D417/14;C07D471/08;C07K5/04;(IPC1-7):A61K31/541;A61K31/537;A61K31/495;A61K31/496;C07D417/02;C07D413/02;C0743/02 主分类号 C07D277/04
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