发明名称 Process for preparing highly functionalized gamma-butyrolactams and gamma-amino acids
摘要 The invention relates to a process for preparing highly functionalized gamma-butyrolactams and gamma-amino acids by reductive amination of mucohalic acid or its derivatives, and discloses a process for preparing pregabalin, a GABA analog with desirable medicinal activity.
申请公布号 US2003225149(A1) 申请公布日期 2003.12.04
申请号 US20030365430 申请日期 2003.02.13
申请人 BLAZECKA PETER G.;DAVIDSON JAMES GUY;ZHANG JI 发明人 BLAZECKA PETER G.;DAVIDSON JAMES GUY;ZHANG JI
分类号 C07D207/38;A61K31/198;A61K31/405;A61K31/4172;C07B61/00;C07C227/12;C07C227/22;C07C229/00;C07C229/04;C07C229/06;C07C229/08;C07C229/28;C07C229/34;C07C229/38;C07D207/24;C07D209/18;C07D213/55;C07D233/66;(IPC1-7):A61K31/417 主分类号 C07D207/38
代理机构 代理人
主权项
地址