发明名称 |
Process for preparing highly functionalized gamma-butyrolactams and gamma-amino acids |
摘要 |
The invention relates to a process for preparing highly functionalized gamma-butyrolactams and gamma-amino acids by reductive amination of mucohalic acid or its derivatives, and discloses a process for preparing pregabalin, a GABA analog with desirable medicinal activity.
|
申请公布号 |
US2003225149(A1) |
申请公布日期 |
2003.12.04 |
申请号 |
US20030365430 |
申请日期 |
2003.02.13 |
申请人 |
BLAZECKA PETER G.;DAVIDSON JAMES GUY;ZHANG JI |
发明人 |
BLAZECKA PETER G.;DAVIDSON JAMES GUY;ZHANG JI |
分类号 |
C07D207/38;A61K31/198;A61K31/405;A61K31/4172;C07B61/00;C07C227/12;C07C227/22;C07C229/00;C07C229/04;C07C229/06;C07C229/08;C07C229/28;C07C229/34;C07C229/38;C07D207/24;C07D209/18;C07D213/55;C07D233/66;(IPC1-7):A61K31/417 |
主分类号 |
C07D207/38 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|