发明名称 Substituted pyrazoles as p38 kinase inhibitors and tumour necrosis factors
摘要 A class of pyrazole derivatives of formula (IB) that are useful for treating p38 kinase mediated disorders are disclosed, wherein R1, R2, R3 and R4 are as described in the specification.
申请公布号 NZ512344(A) 申请公布日期 2003.11.28
申请号 NZ19990512344 申请日期 1999.11.17
申请人 G 发明人 XU, XIANGDONG;YU, YI;RAO, SHASHIDHAR N;SELNESS,SHAUN RAJ;SOUTH, MICHAEL S;STEALEY, MICHAEL A;TALLEY,JOHN JEFFREY;VAZQUEZ, MICHAEL L;WEIER, RICHARD M;HANSON,GUNNAR J;HARTMANN, SUSAN J;HEPPERLE, MICHAEL;HUANG, HE;HANNA, ISH K;KOSZYK, FRANCIS J;LIAO, SHUYUAN;METZ,SUZANNE;PARTIS, RICHARD A;PERRY, THAO D;ANANTANARAYAN,ASHOK;CLARE, MICHAEL;COLLINS, PAUL W;CRICH, JOYCE Z;EVRAJ, RAJESH;FLYNN, DANIEL L;GENG, LIFENG;GRANETO,MATTHEW J;HANAU E
分类号 A61K31/415;A61K31/44;A61K31/4439;A61K31/445;A61K31/454;A61K31/47;A61K31/496;A61K31/50;A61K31/505;A61K31/506;A61K31/52;A61K31/5377;A61P1/04;A61P9/00;A61P11/00;A61P11/06;A61P13/12;A61P19/00;A61P19/02;A61P19/06;A61P29/00;A61P29/02;A61P43/00;C07D401/04;C07D401/14;C07D403/04;C07D403/14;C07D405/14;C07D409/14;C07D413/14;C07D417/14;C07D453/02;C07D471/04;C07D473/00;C07D487/04;(IPC1-7):C07D471/04 主分类号 A61K31/415
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