发明名称 Glucagon antagonists/inverse agonists
摘要 A novel class of compounds, which act to antagonize the action of the glucagon hormone on the glucagon receptor. Owing to their antagonizing effect of the glucagon receptor the compounds may be suitable for the treatment and/or prevention of any glucagon-mediated conditions and diseases such as hyperglycemia, Type 1 diabetes, Type 2 diabetes and obesity.
申请公布号 US2003220350(A1) 申请公布日期 2003.11.27
申请号 US20020233851 申请日期 2002.08.30
申请人 LAU JESPER;MADSEN PETER;SAMS CHRISTIAN;BEHRENS CARSTEN;VAGNER JOSEF;CHRISTENSEN INGE THOGER;LUNDT BEHREND FREDERIK;SIDELMANN ULLA GROVE;THOGERSEN HENNING;LING ANTHONY L.;PLEWE MICHAEL BRUNO;TRUESDALE LARRY KENNETH;JOGENSEN ANKER STEEN;KODRA JANOS TIBOR;SHI SHENGHUA 发明人 LAU JESPER;MADSEN PETER;SAMS CHRISTIAN;BEHRENS CARSTEN;VAGNER JOSEF;CHRISTENSEN INGE THOGER;LUNDT BEHREND FREDERIK;SIDELMANN ULLA GROVE;THOGERSEN HENNING;LING ANTHONY L.;PLEWE MICHAEL BRUNO;TRUESDALE LARRY KENNETH;JOGENSEN ANKER STEEN;KODRA JANOS TIBOR;SHI SHENGHUA
分类号 C07C237/36;C07C237/42;C07C243/38;C07C271/56;C07C271/58;C07C275/24;C07C275/26;C07C275/28;C07C275/30;C07C275/34;C07C275/36;C07C275/38;C07C275/42;C07C275/60;C07C275/62;C07C311/47;C07C317/22;C07C317/32;C07C317/42;C07C323/21;C07C323/44;C07D209/08;C07D209/48;C07D211/58;C07D213/75;C07D215/38;C07D231/40;C07D235/30;C07D257/06;C07D277/72;C07D295/13;C07D295/135;C07D307/68;C07D317/66;C07D319/18;C07D319/20;C07D333/20;C07D333/38;C07D333/60;C07D333/68;C07D333/70;C07D409/12;C07D417/12;C07D487/04;(IPC1-7):A61K31/519;A61K31/41;A61K31/275;A61K31/335 主分类号 C07C237/36
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