发明名称 |
SUBSTITUTED QUINOLONE CARBOXYLIC ACIDS, THEIR DERIVATIVES, SITE OF ACTION, AND USES THEREOF |
摘要 |
Substituted quinolone carboxylic acids and their derivatives are described. These compounds modulate the effect of .gamma.-aminobutyric acid (GABA) via a novel site on the GABAA receptor complex in a therapeutically relevant fashi on and may be used to ameliorate CNS disorders amenable to modulation of the GABAA receptor complex.
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申请公布号 |
CA2484308(A1) |
申请公布日期 |
2003.11.27 |
申请号 |
CA20032484308 |
申请日期 |
2003.05.12 |
申请人 |
THE REGENTS OF THE UNIVERSITY OF CALIFORNIA |
发明人 |
HOGENKAMP, DERK J.;JOHNSTONE, TIMOTHY B.C.;GEE, KELVIN W. |
分类号 |
A61K31/47;A61K31/4709;A61P21/02;A61P25/00;A61P25/02;A61P25/06;A61P25/08;A61P25/18;A61P25/20;A61P25/22;A61P25/24;A61P25/28;A61P25/30;A61P25/36;A61P29/00;A61P43/00;C07D215/56;C07D401/12;(IPC1-7):C07D215/38;C07D215/16;C07D215/20 |
主分类号 |
A61K31/47 |
代理机构 |
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地址 |
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