发明名称 POLYMER PRECURSORS OF RADIOLABELED COMPOUNDS, AND METHODS OF MAKING AND USING THE SAME
摘要 <p>A polymer precursor compound represented by 1: €ƒ€ƒ€ƒ€ƒ€ƒ€ƒ€ƒ€ƒPoly--L---R----Y wherein: Poly represents a polymer; L is selected from: R represents polycyclic aryl or heteroaryl; Y represents hydrogen, alkyl, alkoxyl, carbonyl, formyl, amido, amino, alkylamino, dialkylamino, carboxamido, acylamino, (heterocyclcyl)acylamino, alkylcarboxyamido, C(O)-R 4 , or C(O)NH-R 4 ; R 3 represents independently for each occurrence alkyl, alkenyl or alkynyl; R 4 represents hydrogen, alkyl, alkenyl, heteroalkyl, cycloalkyl, heterocycloalkyl, aryl, heteroaryl, aralkyl, heteroaralkyl, peptide, protein, amino acid, antibody, nucleotide, nucleoside, or -(CH 2 ) m -R 80 ; R 80 represents independently for each occurrence aryl, cycloalkyl, cycloalkenyl, heterocyclyl, or polycyclyl; and m is an integer in the range 0 to 8 inclusive. The polymer precursor is used for preparing radiolabeled compounds.</p>
申请公布号 EP1363954(A2) 申请公布日期 2003.11.26
申请号 EP20020727956 申请日期 2002.03.04
申请人 UNIVERSITY OF WESTERN ONTARIO 发明人 HUNTER, DUNCAN, H.;JANABI, MUSTAFA
分类号 A61K51/06;G01N33/60;C07B59/00;C07C231/12;C07C233/78;C07F7/22;C07K1/04;C07K14/00;C08F2/00;C08F8/00;C08F8/32;C08F8/42;(IPC1-7):C08F8/06 主分类号 A61K51/06
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