发明名称 INHIBITORS OF HISTONE DEACETYLASE
摘要 The invention relates to the inhibition of histone deacetylase. The invention provides compounds e.g. (1) and methods for inhibiting deacetylase enzymatic activity. The invention also provides compositions and methods for treating cell proliferative diseases and conditions. (formula 1). All definitions are as the application.
申请公布号 WO03024448(A3) 申请公布日期 2003.11.13
申请号 WO2002US29017 申请日期 2002.09.12
申请人 METHYLGENE, INC.;DELORME, DANIEL;WOO, SOON, HYUNG;VAISBURG, ARKADII;MORADEL, OSCAR;LEIT, SILVANA;RAEPPEL, STEPHANE;FRECHETTE, SYLVIE;BOUCHAIN, GILIANE 发明人 DELORME, DANIEL;WOO, SOON, HYUNG;VAISBURG, ARKADII;MORADEL, OSCAR;LEIT, SILVANA;RAEPPEL, STEPHANE;FRECHETTE, SYLVIE;BOUCHAIN, GILIANE
分类号 C07D251/46;A61K31/167;A61K31/17;A61K31/18;A61K31/277;A61K31/34;A61K31/343;A61K31/352;A61K31/357;A61K31/36;A61K31/381;A61K31/4035;A61K31/4045;A61K31/407;A61K31/41;A61K31/415;A61K31/4164;A61K31/4184;A61K31/421;A61K31/423;A61K31/4245;A61K31/426;A61K31/428;A61K31/437;A61K31/44;A61K31/4402;A61K31/4406;A61K31/4409;A61K31/4418;A61K31/4436;A61K31/4439;A61K31/444;A61K31/454;A61K31/455;A61K31/47;A61K31/4709;A61K31/472;A61K31/495;A61K31/496;A61P35/00;A61P43/00;C07C233/44;C07C233/80;C07C235/38;C07C235/42;C07C235/56;C07C235/82;C07C235/84;C07C237/20;C07C237/22;C07C237/40;C07C237/42;C07C255/58;C07C255/59;C07C275/34;C07C275/36;C07C311/42;C07C323/32;C07C323/36;C07C323/44;C07C323/60;C07C381/00;C07D209/14;C07D209/46;C07D211/88;C07D213/30;C07D213/38;C07D213/44;C07D213/56;C07D213/70;C07D213/74;C07D213/75;C07D213/81;C07D213/82;C07D213/85;C07D215/22;C07D215/36;C07D215/38;C07D215/48;C07D217/04;C07D231/12;C07D231/38;C07D233/54;C07D233/64;C07D233/84;C07D235/26;C07D235/28;C07D235/30;C07D239/36;C07D239/42;C07D239/47;C07D239/52;C07D239/91;C07D239/96;C07D251/18;C07D251/48;C07D251/50;C07D251/52;C07D251/54;C07D251/70;C07D251/72;C07D253/08;C07D257/04;C07D263/14;C07D263/22;C07D263/24;C07D263/58;C07D265/26;C07D265/36;C07D271/06;C07D271/10;C07D277/20;C07D277/30;C07D277/42;C07D277/70;C07D277/74;C07D277/82;C07D279/16;C07D295/12;C07D295/14;C07D295/155;C07D307/12;C07D307/16;C07D307/28;C07D307/85;C07D311/04;C07D311/22;C07D311/56;C07D311/58;C07D311/74;C07D317/66;C07D319/18;C07D319/20;C07D333/20;C07D333/36;C07D333/38;C07D333/70;C07D401/04;C07D401/12;C07D403/04;C07D405/12;C07D409/12;C07D413/12;C07D417/12;C07D473/16;C07D473/34;C07D473/40;C07D487/04;C07D491/113;C07D495/04;C07D498/04;C07D513/04;C07D521/00;C07F7/08;C07F7/10;C07F7/18;C12N9/99 主分类号 C07D251/46
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