发明名称 COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES
摘要 Disclosed are novel cathepsin S, K, F, L and B reversible inhibitory compounds of the formulas (Ia) and (Ib) where R1, R2, R3, R4, R5, R6, R8, R9 and X aredefined herein. The compoundsare useful for treating autoimmune and other diseases. Also disclosed are processes for making such novel compounds.
申请公布号 WO03029200(A3) 申请公布日期 2003.11.13
申请号 WO2002US30644 申请日期 2002.09.27
申请人 BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 发明人 BEKKALI, YOUNES;HICKEY, EUGENE, R.;WEIMIN, LIU;PATEL, USHA, R.;SPERO, DENICE, MARY;SUN, SANXING;THOMSON, DAVID, S.;WARD, YANCEY, D.;YOUNG, ERICK, R., R.
分类号 C07D295/12;A61K31/277;A61K31/341;A61K31/351;A61K31/428;A61K31/517;A61K31/536;A61K31/5375;A61K31/5377;A61P1/04;A61P3/10;A61P5/14;A61P9/10;A61P11/06;A61P13/12;A61P15/00;A61P17/00;A61P17/06;A61P19/02;A61P19/10;A61P21/04;A61P25/00;A61P25/28;A61P29/00;A61P37/00;A61P37/02;A61P37/06;A61P43/00;C07C257/20;C07C269/06;C07C271/20;C07C271/64;C07C319/20;C07C323/41;C07C323/60;C07D211/22;C07D213/30;C07D213/57;C07D239/80;C07D263/32;C07D265/24;C07D275/06;C07D277/30;C07D295/14;C07D295/215;C07D307/12;C07D307/54;C07D309/08;C07D309/12;C07D333/24;C07D401/04;C07D401/06 主分类号 C07D295/12
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