发明名称 OXAZOLIDINONE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS BASED ON THEREOF
摘要 FIELD: organic chemistry, pharmacy. SUBSTANCE: invention relates to novel oxazolidinone derivatives of the formula (I) , their enantiomers or their pharmaceutically acceptable salts wherein R means hydrogen atom or C1-6-alkyl optionally substituted with group taken among cyano-, fluorine, chlorine atom, hydroxy- or carbamoyl; R1 and R2 represent independently fluorine or hydrogen atom; R3 represents C1-6-alkyl; X represents oxygen or sulfur atom. Invention relates to pharmaceutical compositions eliciting an antibacterial effect and containing compound of the formula (I) as an active component and pharmaceutically acceptable carrier. Invention provides preparing the novel compound eliciting an antibacterial effect. EFFECT: valuable medicinal property of derivatives. 8 cl, 1 tbl, 5 ex
申请公布号 RU2215740(C2) 申请公布日期 2003.11.10
申请号 RU20000114891 申请日期 1998.10.30
申请人 FARMATSIJA EHND APDZHON KOMPANI 发明人 KHESTER DZHEKSON B. ML.
分类号 A61K31/422;A61K31/551;A61P31/00;A61P31/04;C07D243/00;C07D263/00;C07D413/10;C07D413/14;(IPC1-7):C07D413/10 主分类号 A61K31/422
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