发明名称 Process for the preparation of basic antibiotic inorganic acid addition salts and oxalate intermediate
摘要 A production process which comprises subjecting a basic antibiotic.oxalate (II) to salt-exchange with an alkali earth metal salt (III) of an inorganic acid:wherein the ring A means the basic antibiotic; R<10 >means a protected functional group used in organic synthesis; Ak-E means the alkali earth metal; and B means the inorganic acid, respectively.
申请公布号 US6642377(B1) 申请公布日期 2003.11.04
申请号 US20020030909 申请日期 2002.01.14
申请人 EISAI CO., LTD. 发明人 KAYANO AKIO;CHIBA HIROYUKI;NAKAMURA TAIJU;SAKURAI SHIN;ISHIZUKA HIROYUKI;SAITO HIROYUKI;KOMATSU YUUKI;SASHO MANABU;SATO NOBUAKI;NEGI SHIGETO
分类号 C07D477/02;C07D477/08;C07D477/20;C07D499/68;C07D501/22;C07D501/36;C07D501/46;(IPC1-7):C07D477/20 主分类号 C07D477/02
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