发明名称 PROCESS FOR PREPARING HETEROARYL AND UNSATURATED HETEROCYCLOALKYLMAGNESIUM REAGENTS AND USES
摘要 The present invention is directed to a novel process for preparing heteroaryl and unsaturated heterocycloalkylmagnesium reagents that are useful in the synthesis of a variety of pharmaceuticals, in particular certain cysteine protease inhibitors.
申请公布号 WO03087068(A1) 申请公布日期 2003.10.23
申请号 WO2003US12279 申请日期 2003.04.16
申请人 AXYS PHARMACEUTICALS, INC.;AVENTIS PHARMACEUTICALS, INC.;LI, JIAYAO;LINK, JOHN, O.;COLLADANT, COLETTE 发明人 LI, JIAYAO;LINK, JOHN, O.;COLLADANT, COLETTE
分类号 C07D263/56;C07D277/64;C07D498/04;C07F3/02;(IPC1-7):C07D263/52;C07D413/12 主分类号 C07D263/56
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