发明名称 |
INHIBITORS AGAINST THE PRODUCTION AND RELEASE OF INFLAMMATORY CYTOKINES |
摘要 |
A medicament having inhibitory activity against NF- kappa B activation, which comprises a compound represented by the following general formula (I) or a pharmacologically acceptable salt as an active ingredient: <CHEM> wherein X represents a connecting group, A represents hydrogen atom or acetyl group, E represents an aryl group or a heteroaryl group, and ring X represents an arene or a heteroarene.
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申请公布号 |
EP1352650(A1) |
申请公布日期 |
2003.10.15 |
申请号 |
EP20010271124 |
申请日期 |
2001.12.18 |
申请人 |
INSTITUTE OF MEDICINAL MOLECULAR DESIGN, INC. |
发明人 |
MUTO, SUSUMU;NAGANO, TATSUO;SAOTOME, TOMOMI;ITAI, AKIKO |
分类号 |
A61K31/055;A61K31/12;A61K31/136;A61K31/166;A61K31/167;A61K31/17;A61K31/18;A61K31/357;A61K31/403;A61K31/404;A61K31/415;A61K31/421;A61K31/422;A61K31/428;A61K31/433;A61K31/44;A61K31/47;A61K31/498;A61K31/505;A61K31/5375;A61K31/695;A61P29/00;C07D207/32;C07D207/327;C07D209/08;C07D209/34;C07D209/42;C07D209/80;C07D209/88;C07D213/64;C07D213/65;C07D213/75;C07D215/12;C07D215/38;C07D231/40;C07D239/22;C07D241/44;C07D263/48;C07D277/24;C07D285/08;C07D321/10;C07D333/16;C07D333/38;C07D413/14;C07D471/04;(IPC1-7):A61K31/055;A61K31/537 |
主分类号 |
A61K31/055 |
代理机构 |
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代理人 |
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地址 |
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