发明名称 |
PROCESS FOR PREPARING ACTIVE ESTERS |
摘要 |
<p>The present invention relates to a method for the preparation of active ester, characterized by subjecting to a reaction a mixture of a carboxylic acid, which is a starting material, reagent which forms active ester and a base or a starting material carboxylic acid. <??>The present invention provides an active ester useful as an intermediate of pharmaceutical drugs etc. in high yield using an inexpensive reagent, in one-pot reaction, without causing isomerization, regardless of the structure of starting material carboxylic acid.</p> |
申请公布号 |
EP1350790(A1) |
申请公布日期 |
2003.10.08 |
申请号 |
EP20010270527 |
申请日期 |
2001.12.13 |
申请人 |
ONO PHARMACEUTICAL CO., LTD. |
发明人 |
OKUYAMA, SHIGEHIRO;MASAOKA, HIDEO |
分类号 |
C07D207/46;C07D417/12;(IPC1-7):C07D207/46;C07B41/12;C07B43/00 |
主分类号 |
C07D207/46 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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