发明名称 5-amino-benzofuran-2-carboxylsyrederivater
摘要 <p>5-(Amino or piperazino)-benzofuran-2-carboxamides (I) are new. 5-(Amino or piperazino)-benzofuran-2-carboxamides of formula (I) and their salts are new. R1 = NH2, or piperazino; R2 = H, Cl, Br, OH, or OA; X = CONR4R5, or CO-Het; R4, R5 = H, A, or benzyl; A = 1-4C alkyl; and Het = imidazol-1-yl, triazol-1-yl or tetrazol-1-yl. An Independent claim is also included for the preparation of (I).</p>
申请公布号 DK0738722(T3) 申请公布日期 2003.09.29
申请号 DK19960105701T 申请日期 1996.04.11
申请人 MERCK PATENT GMBH 发明人 BOETTCHER, HENNING, DR.;BATHE, ANDREAS, DR.;HELFERT, BERND;SCHUSTER, KURT
分类号 C07D307/81;A61K31/34;A61K31/343;A61K31/40;A61K31/415;A61K31/495;A61K31/50;A61P25/00;C07D307/85;C07D405/04;C07D405/06;C07D405/12;(IPC1-7):C07D307/85 主分类号 C07D307/81
代理机构 代理人
主权项
地址