发明名称 |
5-(2-substituted-5-heterocyclylsulphonylpyrid-3-YL)- dihydropyrazolo[4,3-d]pyrimidin-7-ones as phosphodiesterase inhibitors |
摘要 |
Compounds of formula (I), which are useful in the curative and prophylactic treatment of a medical condition for which inhibition of a cyclic guanosine 3',5'- monophosphate phosphodiesterase (e.g. cGMP PDE5) and having utility in therapeutic areas such as erectile male dysfunction (MED) are disclosed, wherein R1, R2, R3, R4 and X are as described in the specification. |
申请公布号 |
NZ517324(A) |
申请公布日期 |
2003.09.26 |
申请号 |
NZ20000517324 |
申请日期 |
2000.10.04 |
申请人 |
PFIZER, INC |
发明人 |
ALLERTON, CHARLOTTE MOIRA NORFOR;BARBER, CHRISTOPHERGORDON;MAW, GRAHAM NIGEL;RAWSON, DAVID JAMES |
分类号 |
A61K;A61K31/519;A61K31/5377;A61P;A61P15/00;A61P15/08;A61P15/10;A61P15/12;C07D;C07D487/04 |
主分类号 |
A61K |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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