发明名称 Method for producing delta-aminopentadienoate derivatives
摘要 The invention is a method for producing delta-aminopentadienoate derivatives of formula (1), the method comprising reacting a streptocyanine derivative of formula (2) with an ester derivative of formula (3) in the presence of an organic base. In formulae (1) to (3), R<1 >represents an alkyl group or an aryl group; R<2>, R<3>, R<4 >and R<5 >independently represent a hydrogen atom or an alkyl group; R<2 >and R<3>, or R<4 >and R<5 >may bond to each other to form a ring; Y represents an electron attractive group; X represents an acid radical; n indicates 0 or a positive number, which is no more than 5; Y may bond to R<1 >to form a ring.
申请公布号 US2003181483(A1) 申请公布日期 2003.09.25
申请号 US20030395166 申请日期 2003.03.25
申请人 IKEGAWA AKIHIKO;MOTOKI MASUJI;YAMAKAWA KATSUYOSHI 发明人 IKEGAWA AKIHIKO;MOTOKI MASUJI;YAMAKAWA KATSUYOSHI
分类号 C07B61/00;C07C227/02;C07C315/04;C07C317/48;(IPC1-7):A61K31/445;A61K31/40;A61K31/22;C07D211/20 主分类号 C07B61/00
代理机构 代理人
主权项
地址