发明名称 |
Fremgangsmåte for fremstilling av imidazol-forbindelser |
摘要 |
A process for the preparation of 4-(3-chlorophenyl)-6-[(4-chlorophenyl)hydroxy(1-methyl-1H-imidazol-5-yl)methyl]-1-methyl-2(1H)-quinolinone which comprises reacting 6-(4-chlorobenzoyl)-4-(3-chlorophenyl)-1-methyl-2(1H)-quinolinone with a C6-8alkyllithium compound, 1-methylimidazole and a tri(C4-6alkyl)silyl halide to obtain better yields of the above product. |
申请公布号 |
NO20034003(D0) |
申请公布日期 |
2003.09.10 |
申请号 |
NO20030004003 |
申请日期 |
2003.09.10 |
申请人 |
JANSSEN PHARMACEUTICA NV |
发明人 |
FILLIERS, WALTER FERDINAND MARIA;BROECKX, RUDY LAURENT MARIA;LEURS, STEFAN MARCEL HERMAN |
分类号 |
A61K31/4709;A61P35/00;C07D401/06;C07D403/06;(IPC1-7):C07D |
主分类号 |
A61K31/4709 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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