发明名称 Indolylpiperidine derivatives as antihistaminic and antiallergic agents
摘要 A compound of formula (I), wherein: A1 represents an alkylene, alkyleneoxy, alkylenethio, alkanoyl or hydroxyalkylene group, A2 represents a single bond, an alkylene or alkenylene group, W represents a single bond or an optionally substituted phenylene or furanylene group, R1 represents a hydrogen, alkyl, alkenyl, alkynyl, alkoxyalkyl, alkenyloxyalkyl, alkynyloxyalkyl, alkoxy-alkoxyalkyl, or an optionally substituted phenylalkyl group, R2 represents a hydrogen, halogen, alkyl or alkoxy group, and R3 represents a carboxyl or tetrazolyl group. The compounds are used in the preparation of medicaments for use as antihistaminic or antiallergic agents.
申请公布号 NZ515649(A) 申请公布日期 2003.08.29
申请号 NZ20000515649 申请日期 2000.05.31
申请人 ALMIRALL PRODESFARMA, S 发明人 PAGES SANTACANA, LLUIS;FONQUERNA POU, SILVIA;PUIG DURAN, CARLES;FERNANDEZ FORNER, DOLORS
分类号 A61K31/445;A61K31/4525;A61K31/454;A61P11/02;A61P11/04;A61P11/06;A61P27/02;A61P37/08;C07D401/04;C07D401/14;C07D405/14;(IPC1-7):C07D401/04 主分类号 A61K31/445
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