发明名称 |
CONTROLLED SYNTHESIS OF ZIPRASIDONE AND COMPOSITIONS THEREOF |
摘要 |
The subject invention provides a ziprasidone composition that comprises not greater than 1000 ppm des-chloro ziprasidone, preferably not greater than about 500 ppm des-chloro ziprasidone, and more preferably not greater than about 100 ppm des-chloro ziprasidone. Methods for synthesizing and using such ziprasidone compositions are also provided.
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申请公布号 |
WO03070246(A1) |
申请公布日期 |
2003.08.28 |
申请号 |
WO2003IB00642 |
申请日期 |
2003.02.17 |
申请人 |
PFIZER PRODUCTS INC. |
发明人 |
BUSCH, FRANK, ROBERT;GROBIN, ADAM, WORTH;HOWARD, HARRY, RALPH, JR.;LEEMAN, KYLE, ROBERT |
分类号 |
C07D417/12;A61K;A61K31/496;A61P;A61P25/00;A61P25/06;A61P25/14;A61P25/22;A61P25/28;A61P27/06;(IPC1-7):A61K31/496 |
主分类号 |
C07D417/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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