摘要 |
4'-C-Cyano-2'-deoxypurine nucleosides represented by the following general formula [I] which have an excellent anti-HIV effect, in particular, an efficacy on multidrug-resistant HIV strains having resistance to a plural number of anti-HIV drugs such as AZT, ddI, ddC, d4T and 3TC without causing any problems in cytotoxicity; and medicinal compositions comprising such a compound and a pharmaceutically acceptable carrier: [I] wherein B represents a purine base; and R represents hydrogen or phosphate.
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申请人 |
YAMASA CORPORATION;KOHGO, SATORU;YAMADA, KOHEI;SAKATA, SHINJI;OHRUI, HIROSHI;KODAMA, EIICHI;MATSUOKA, MASAO;MITSUYA, HIROAKI |
发明人 |
KOHGO, SATORU;YAMADA, KOHEI;SAKATA, SHINJI;OHRUI, HIROSHI;KODAMA, EIICHI;MATSUOKA, MASAO;MITSUYA, HIROAKI |