发明名称 |
Fused azabicyclic compounds that inhibit vanilloid receptor subtype 1 (VR1) receptor |
摘要 |
Compounds of formula (I) are novel VR1 antagonists that are useful in treating pain, inflammatory thermal hyperalgesia, urinary incontinence and bladder overactivity.
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申请公布号 |
US2003158188(A1) |
申请公布日期 |
2003.08.21 |
申请号 |
US20020079324 |
申请日期 |
2002.02.20 |
申请人 |
LEE CHIH-HUNG;BAYBURT EROL K.;DIDOMENICO STANLEY;DRIZIN IRENE;GOMTSYAN ARTHUR R.;KOENIG JOHN R.;PERNER RICHARD J.;SCHMIDT ROBERT G.;TURNER SEAN C.;WHITE TAMMIE K.;ZHENG GUO ZHU |
发明人 |
LEE CHIH-HUNG;BAYBURT EROL K.;DIDOMENICO STANLEY;DRIZIN IRENE;GOMTSYAN ARTHUR R.;KOENIG JOHN R.;PERNER RICHARD J.;SCHMIDT ROBERT G.;TURNER SEAN C.;WHITE TAMMIE K.;ZHENG GUO ZHU |
分类号 |
A61K31/404;A61K31/416;A61K31/47;A61K31/472;A61K31/496;A61K31/5377;A61K31/541;C07D209/08;C07D217/02;C07D217/26;C07D231/56;C07D237/28;C07D405/12;(IPC1-7):A61K31/541;A61K31/537;C07D417/02;C07D413/02;C0743/02 |
主分类号 |
A61K31/404 |
代理机构 |
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地址 |
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