发明名称 Fused azabicyclic compounds that inhibit vanilloid receptor subtype 1 (VR1) receptor
摘要 Compounds of formula (I) are novel VR1 antagonists that are useful in treating pain, inflammatory thermal hyperalgesia, urinary incontinence and bladder overactivity.
申请公布号 US2003158188(A1) 申请公布日期 2003.08.21
申请号 US20020079324 申请日期 2002.02.20
申请人 LEE CHIH-HUNG;BAYBURT EROL K.;DIDOMENICO STANLEY;DRIZIN IRENE;GOMTSYAN ARTHUR R.;KOENIG JOHN R.;PERNER RICHARD J.;SCHMIDT ROBERT G.;TURNER SEAN C.;WHITE TAMMIE K.;ZHENG GUO ZHU 发明人 LEE CHIH-HUNG;BAYBURT EROL K.;DIDOMENICO STANLEY;DRIZIN IRENE;GOMTSYAN ARTHUR R.;KOENIG JOHN R.;PERNER RICHARD J.;SCHMIDT ROBERT G.;TURNER SEAN C.;WHITE TAMMIE K.;ZHENG GUO ZHU
分类号 A61K31/404;A61K31/416;A61K31/47;A61K31/472;A61K31/496;A61K31/5377;A61K31/541;C07D209/08;C07D217/02;C07D217/26;C07D231/56;C07D237/28;C07D405/12;(IPC1-7):A61K31/541;A61K31/537;C07D417/02;C07D413/02;C0743/02 主分类号 A61K31/404
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