发明名称 |
SUBSTITUTED PHENOL DERIVATIVES OR SALTS THEREOF AS INHIBITORS OF COAGULATION FACTOR X |
摘要 |
<p>There are provided compounds having an anticoagulant action on the basis of inhibition of activated blood coagulation factor X and being useful as anticoagulants or preventive/therapeutic agents for diseases induced by thrombosis or embolism. Effective ingredients are the compounds such as 4'-bromo-2'-Ä(5-chloro-2-pyridyl)carbamoyl)-6- beta -D-galactopyranosyloxy-1-isopropylpiperidine-4-carboxanilide, 2'-(2-acetamido-2-deoxy- beta -D-glucopyranosyloxy)-4'-bromo-6'-Ä(5-chloro-2-pyridyl)carbamoylÜ-1-is opropylpiperidine-4-carboxanilide, etc. or salts thereof.</p> |
申请公布号 |
EP1336605(A1) |
申请公布日期 |
2003.08.20 |
申请号 |
EP20010997188 |
申请日期 |
2001.11.21 |
申请人 |
YAMANOUCHI PHARMACEUTICAL CO. LTD. |
发明人 |
ISHIHARA, TSUKASA;HIRAYAMA, FUKUSHI;SUGASAWA, KEIZO;KOGA, YUJI;KADOKURA, TAKESHI;SHIGENAGA, TAKESHI |
分类号 |
C07D401/12;A61P7/02;A61P9/10;C07D211/26;C07D401/14;C07H15/203;C07H15/26;(IPC1-7):C07D211/26;A61K31/454;A61K31/445;A61K31/706;C07D405/12;C07D405/14;C07D413/12;C07D417/12;A61K31/506;A61K31/551;A61K31/705;A61K31/501 |
主分类号 |
C07D401/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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