发明名称 |
Xanthine derivatives intended for preparing a medicament used for the treatment and prophylaxis of shock diseases, novel xanthine derivatives, and process of their preparation |
摘要 |
<p>Slou eniny obecn ho vzorce I, ve kter²ch R.sup.1.n. je (C.sub.1.n.-C.sub.5.n.)-alkyl, (C.sub.1.n.-C.sub.2.n.)-alkoxy- (C.sub.1.n.-C.sub.3.n.)-alkyl nebo pop° pad halogen substituovan² fenyl i fenyl-(C.sub.1.n.-C.sub.2.n.)-alkyl, A je (C.sub.1.n.-C.sub.4.n.)-alkylen, a R.sup.2.n. je (C.sub.1.n.-C.sub.5.n.)-alkyl, (C.sub.3.n.-C.sub.6.n.)-cykloalkyl, (C.sub.4.n.-C.sub.8.n.)-cykloalkylalkyl, fenyl nebo fenyl-(C.sub.1.n.-C.sub.2.n.)-alkyl jsou vhodn k p° prav l iv k l en a profylaxi Üokov²ch onemocn n . Zp sob jejich p° pravy a meziprodukty v jejich p° prav obecn ho vzorce VIII, ve kter m R.sup.a.n. je benzyl./</p> |
申请公布号 |
CZ292205(B6) |
申请公布日期 |
2003.08.13 |
申请号 |
CZ19970001743 |
申请日期 |
1997.06.05 |
申请人 |
HOECHST AKTIENGESELLSCHAFT |
发明人 |
GEBERT ULRICH DR.;WOLF ERHARD DR.;DEFOSSA ELISABETH DR.;HEINELT UWE DR.;ANAGNOSTOPULOS HIRISTO DB.;RUDOLPHI KARL DR.;GROME JOHN J. DR. |
分类号 |
C07D473/04;A61K31/505;A61K31/522;A61P7/08;A61P9/00;A61P9/10;A61P31/04;A61P31/12;A61P43/00;C07D473/06;(IPC1-7):C07D473/04 |
主分类号 |
C07D473/04 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|