发明名称 4-SULFIDE / SULFOXIDE / SULFONYL-1H-PYRAZOLYL DERIVATIVE COMPOUNDS, FOR USE IN DISEASES ASSOCIATED WITH THE 5-HT2C RECEPTOR
摘要 Disclosed are 4-sulfide / sulfoxide / sulfonyl-1<i>H</i>-pyrazolyl derivative compounds of formulas (I) or (II):wherein the variables n, R, R<sb>1</sb>, R<sb>2</sb>, R<sb>3</sb>, R<sb>3'</sb>, R<sb>4</sb>, R<sb>4'</sb>, R<sb>5</sb> and R<sb>6</sb> are as defined in the specification. The compounds are useful for the treatment or prevention of diseases and/or behaviors involving the 5-HT<sb>2C</sb> receptor.
申请公布号 WO03057674(A1) 申请公布日期 2003.07.17
申请号 WO2002US41635 申请日期 2002.12.28
申请人 BAYER CORPORATION;LADOUCEUR, GAETAN, H.;VELTHUISEN, EMIL;CHOI, SOONGYOU;ZHANG, ZHONGHUA;WANG, YAMIN;BARYZA, JEREMY, L.;COISH, PHILIP;SMITH, ROGER;CHEN, MICHAEL 发明人 LADOUCEUR, GAETAN, H.;VELTHUISEN, EMIL;CHOI, SOONGYOU;ZHANG, ZHONGHUA;WANG, YAMIN;BARYZA, JEREMY, L.;COISH, PHILIP;SMITH, ROGER;CHEN, MICHAEL
分类号 A61K31/415;A61K31/4152;A61K31/4155;A61K31/423;A61K31/427;A61K31/428;A61K31/4439;A61K31/454;A61K31/506;A61K31/5377;A61P3/04;A61P3/10;A61P15/12;A61P25/00;A61P43/00;C07D231/18;C07D401/12;C07D403/04;C07D403/12;C07D405/12;C07D413/12;C07D417/12;(IPC1-7):C07D231/18 主分类号 A61K31/415
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