发明名称 THIENOPYRIMIDINE COMPOUNDS AS PROTEIN TYROSINE KINASE INHIBITORS
摘要 The present invention relates to thienopyrmidine compounds of formula (I) (one of A<sp>1 </sp>and A<sp>2 </sp>is S and the other is CH), salts thereof, as well as use and preparation of the same. These compounds are inhibitors of various protein tyrosine kinases (PTKs) of the ErbB family and consequently are useful in the treatment of disorders mediated by aberrant activity of such kinases.
申请公布号 WO03053446(A1) 申请公布日期 2003.07.03
申请号 WO2002US39872 申请日期 2002.12.13
申请人 SMITHKLINE BEECHAM CORPORATION;CAFERRO, THOMAS, R;CHAMBERLAIN, STANLEY, DAWES;DONALDSON, KELLY, HORNE;HARRIS, PHILIP, ANTHONY;GAUL, MICHAEL, DAVID;UEHLING, DAVID, EDWARD;VANDERWALL, DANA, EDWARD 发明人 CAFERRO, THOMAS, R;CHAMBERLAIN, STANLEY, DAWES;DONALDSON, KELLY, HORNE;HARRIS, PHILIP, ANTHONY;GAUL, MICHAEL, DAVID;UEHLING, DAVID, EDWARD;VANDERWALL, DANA, EDWARD
分类号 A61K31/337;A61K31/475;A61K31/513;A61K31/519;A61K31/5377;A61K31/541;A61K31/7072;A61K45/00;A61P11/08;A61P17/06;A61P29/00;A61P35/00;A61P43/00;C07D495/04;(IPC1-7):A61K31/519 主分类号 A61K31/337
代理机构 代理人
主权项
地址