发明名称 |
Method for the preparation of tetrahydrobenzothiepines |
摘要 |
Among its several embodiments, the present invention provides an improved process for the preparation of tetrahydrobenzothiepine-1,1-dioxide compounds; the provision of a process for preparing a diastereomeric mixture of tetrahydrobenzothiepine-1,1-dioxide compounds from a single diastereomer of such compounds; the provision of a process for the preparation of 3-bromo-2-substituted propionaldehyde compounds; and the provision of a process for the preparation of 3-thio-2-substituted propionaldehyde compounds.
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申请公布号 |
US6586434(B2) |
申请公布日期 |
2003.07.01 |
申请号 |
US20010802279 |
申请日期 |
2001.03.08 |
申请人 |
G.D. SEARLE, LLC |
发明人 |
BABIAK KEVIN A.;CARPENTER ANDREW;CHOU SHINE;COLSON PIERRE-JEAN;FARID PAYMAN;HETT ROBERT;HUBER CHRISTIAN H.;KOELLER KEVIN J.;LAWSON JON P.;LI JAMES;MAR EDUARDO K.;MILLER LAWRENCE M.;ORLOVSKI VLADISLAV;PETERSON JAMES C.;POZZO MARK J.;PRZYBYLA CLAIRE A.;TREMONT SAMUEL J.;TRIVEDI JAY S.;WAGNER GRACE M.;WEISENBURGER GERALD A.;ZHI BENXIN |
分类号 |
C07D317/18;A61K31/235;A61K31/38;A61K31/495;A61K31/4995;A61P3/06;A61P43/00;C07B53/00;C07B55/00;C07B57/00;C07B61/00;C07C201/12;C07C205/35;C07C315/02;C07C315/04;C07C317/24;C07C317/36;C07C319/14;C07C321/28;C07D337/08;C07D409/12;C07D487/08;(IPC1-7):A61K31/495;C07D337/00;C07D487/00 |
主分类号 |
C07D317/18 |
代理机构 |
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代理人 |
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地址 |
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