发明名称 PHOSPHONIC ACID COMPOUNDS AS INHIBITORS OF SERINE PROTEASES
摘要 The present invention is directed to phosphonic acid compounds useful as serine protease inhibitors, compositions thereof and methods for treating inflammatory and serine protease mediated disorders.
申请公布号 CA2464111(A1) 申请公布日期 2003.05.01
申请号 CA20022464111 申请日期 2002.10.17
申请人 ORTHO-MCNEIL PHARMACEUTICAL, INC. 发明人 MARYANOFF, BRUCE E.;QIAN, YUN;HAWKINS, MICHAEL J.;GRECO, MICHAEL N.;ALMOND, HAROLD R.;DE GARAVILLA, LAWRENCE;HUMORA, MICHAEL J.;PATEL, MITUL N.;NILSEN, CHRISTOPHER NORMAN;WALKER, DONALD GILMORE;CESCO-CANCIAN, SERGIO
分类号 A61K31/662;A61P3/06;A61P9/00;A61P9/10;A61P11/00;A61P11/02;A61P11/06;A61P13/12;A61P17/06;A61P19/02;A61P27/02;A61P29/00;A61P37/08;A61P43/00;C07F9/08;C07F9/38;C07F9/40;C07F9/572;C07F9/59;C07F9/6509;C07F9/655;C07F9/6558;C07F9/6561;(IPC1-7):C07F9/08;C07F9/32 主分类号 A61K31/662
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