发明名称 |
Trisubstituted-N-[(1S)-1,2,3,4-terrahydro-1-naphthalenyl]benzamides which inhibit P2X2/3 containing receptors |
摘要 |
Compounds of formula (I) are novel P2X3 and P2X2/P2X3 antagonists which are useful in treating pain, urinary incontinence and bladder overactivity.
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申请公布号 |
US2003083359(A1) |
申请公布日期 |
2003.05.01 |
申请号 |
US20020141989 |
申请日期 |
2002.05.10 |
申请人 |
LEE CHIH-HUNG;PERNER RICHARD J.;LARSON DANIEL P.;KOENIG JOHN R.;GOMTSYAN ARTHUR R.;ZHENG GUO ZHU;DIDOMENICO STANLEY;STEWART ANDREW O.;BAYBURT EROL K. |
发明人 |
LEE CHIH-HUNG;PERNER RICHARD J.;LARSON DANIEL P.;KOENIG JOHN R.;GOMTSYAN ARTHUR R.;ZHENG GUO ZHU;DIDOMENICO STANLEY;STEWART ANDREW O.;BAYBURT EROL K. |
分类号 |
C07D213/40;C07D213/68;C07D213/71;C07D239/34;C07D309/12;C07D317/72;C07D333/20;C07D333/34;C07D333/72;(IPC1-7):C07D409/02;A61K31/443 |
主分类号 |
C07D213/40 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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