发明名称 PHOSPHONIC ACID COMPOUNDS AS INHIBITORS OF SERINE PROTEASES
摘要 The present invention is directed to phosphonic acid compounds useful as serine protease inhibitors, compositions thereof and methods for treating inflammatory and serine protease mediated disorders.
申请公布号 WO03035654(A1) 申请公布日期 2003.05.01
申请号 WO2002US33206 申请日期 2002.10.17
申请人 ORTHO-MCNEIL PHARMACEUTICAL, INC. 发明人 GRECO, MICHAEL, N.;ALMOND, HAROLD, R.;DE GARAVILLA, LAWRENCE;HAWKINS, MICHAEL, J.;MARYANOFF, BRUCE, E.;QIAN, YUN;WALKER, DONALD, GILMORE;CESCO-CANCIAN, SERGIO;NILSEN, CHRISTOPHER, NORMAN;PATEL, MITUL, N.;HUMORA, MICHAEL, J.
分类号 A61K31/662;A61P3/06;A61P9/00;A61P9/10;A61P11/00;A61P11/02;A61P11/06;A61P13/12;A61P17/06;A61P19/02;A61P27/02;A61P29/00;A61P37/08;A61P43/00;C07F9/08;C07F9/38;C07F9/40;C07F9/572;C07F9/59;C07F9/6509;C07F9/655;C07F9/6558;C07F9/6561;(IPC1-7):C07F9/08;C07F9/32 主分类号 A61K31/662
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