发明名称 |
AZOLES CONTAINING ESTERS WITH AMINO ACIDS AS ANTIMYCOTIC FORMS |
摘要 |
The invention relates to compounds with the formula where -A-B- means bivalent radical with the formula -N=CH- (a), -CH=N - (b), -CH=CH- (c), L meaning acyl residue of aminoacid; D is azole containing 1,3- or 1,4-dioxolan derivative. The invention also relates to their N-oxides, pharmaceutically acceptable adjunctive salts and stereochemical isomers, to the preparation of the compounds, to compositions containing them and to their use as wide-spectral antimycotic form. 19 claims |
申请公布号 |
BG63872(B1) |
申请公布日期 |
2003.04.30 |
申请号 |
BG19990103171 |
申请日期 |
1999.02.11 |
申请人 |
JANSSEN PHARMACEUTICA N.V. |
发明人 |
MEERPOEL, LIEVEN;HEERES, JAN;HENDRICKX, ROBERT J. |
分类号 |
C07D405/14;A61K;A61K31/495;A61K31/496;A61P31/10;C07D;C07D521/00;(IPC1-7):C07D405/14 |
主分类号 |
C07D405/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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