发明名称 |
PROCESS FOR THE PREPARATION OF 5-PHENYLPENTANOYL-ALA-ARGL-{2-[3-AMINO-2- OXOPYRROLIDIN-1-YL]PROPIONYL}-ALA-ARG-ALA-4-AMINOPHENYLACETAMIDE |
摘要 |
A process for the preparation of a salt of 5-phenylpentanoyl-(S)-arginyl-(S)-alanyl-{(S)-2-[(R)-3-amino-2-oxopyrrolidin-1-yl]propionyl}-(S)-alanyl-(S)-arginyl-(S)-alanyl-4-aminophenylacetamide (SEQ ID NO: 1) which comprises deprotection of a compound of the formula II or a salt thereof: wherein Pg and R<1 >are defined in the description. Also claimed are intermediates used in the process and the processes for the preparation of the intermediates.
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申请公布号 |
KR20030033001(A) |
申请公布日期 |
2003.04.26 |
申请号 |
KR20037000906 |
申请日期 |
2003.01.21 |
申请人 |
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发明人 |
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分类号 |
C07D207/14;C07K7/02;C07B61/00;C07C231/02;C07C237/20;C07C271/64;C07K5/08;C07K7/06;C07K14/47;C07K14/74 |
主分类号 |
C07D207/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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