发明名称 QUINUCLIDINE DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS M2 AND/OR M3 MUSCARINIC RECEPTOR INHIBITORS
摘要 The invention concerns quinuclidine derivatives of formula I or II wherein the substituents are as defined in the specification, as well as their use as pharmaceuticals. The compounds of the invention_show high affinities for m3 and/or m2 muscarinic receptors and are particularly suited for treating urinary incontinence.
申请公布号 WO03033495(A1) 申请公布日期 2003.04.24
申请号 WO2002EP10644 申请日期 2002.09.23
申请人 UCB, S.A.;GUYAUX, MICHEL;DINESH, CHIMMANAMADA U.;MIOSKOWSKI, CHARLES;QUERE, LUC;STARCK, JEAN-PHILIPPE;TALAGA, PATRICE;WAGNER, ALAIN;ZANDA, MATTEO 发明人 GUYAUX, MICHEL;DINESH, CHIMMANAMADA U.;MIOSKOWSKI, CHARLES;QUERE, LUC;STARCK, JEAN-PHILIPPE;TALAGA, PATRICE;WAGNER, ALAIN;ZANDA, MATTEO
分类号 A61K31/439;A61K31/444;A61P1/00;A61P9/00;A61P11/00;A61P13/02;A61P25/20;A61P25/28;C07D453/02;C07F7/10 主分类号 A61K31/439
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