发明名称 3-[4-(SUBSTITUTED HETEROCYCLYL)-PYRROL-2-YLMETHYLIDENE]-2-INDOLINONE DERIVATIVES AS KINASE INHIBITORS
摘要 The present invention relates to certain 3-[4-(substituted Heterocyclyl)-pyrrol-2-ylmethylidene]-2-Indolinone derivatives that inhibit kinases, in particular VEGFR and/or PDGFR kinases. Pharmaceutical compositions comprising these compounds, methods of treating diseases mediated by kinases utilizing pharmaceutical compositions comprising these compounds, and methods of preparing them are also disclosed.
申请公布号 WO03031438(A1) 申请公布日期 2003.04.17
申请号 WO2002US32354 申请日期 2002.10.10
申请人 SUGEN, INC.;MATTSON, MATTHEW;VOJKOVSKY, TOMAS;LIANG, CONGXIN;TANG, PENG, CHO;GUAN, HUIPING 发明人 MATTSON, MATTHEW;VOJKOVSKY, TOMAS;LIANG, CONGXIN;TANG, PENG, CHO;GUAN, HUIPING
分类号 A61K31/404;A61K31/454;A61K31/4545;A61K31/5377;A61P3/10;A61P9/10;A61P17/06;A61P19/02;A61P25/00;A61P29/00;A61P35/00;A61P35/02;A61P37/02;A61P43/00;C07D401/14;C07D403/06;C07D403/12;C07D403/14;C07D413/14;(IPC1-7):C07D401/14 主分类号 A61K31/404
代理机构 代理人
主权项
地址