发明名称 DERIVATIVES OF ARYLMETHYLAMINE FOR USE AS TRYPTASE INHIBITORS, A PHARMACEUTICAL COMPOSITION BASED THEREON (VARIANTS)
摘要 Provided herein are compounds of formula (I) wherein R1-4, n and Ar are as defined in claim 1, and their pharmaceutical compositions. These compounds are tryptase inhibitors and may be used in the treatment of e.g. asthma and inflammatory diseases.
申请公布号 UA74579(C2) 申请公布日期 2003.04.15
申请号 UA20021210404 申请日期 2001.04.27
申请人 AVENTIS PHARMACEUTICALS INC. 发明人
分类号 A61K31/451;A61K31/452;A61K31/4525;A61K31/453;A61K31/4535;A61K31/454;A61K31/4545;A61K31/4709;A61K31/473;A61K31/496;A61K31/501;A61K31/519;A61K31/537;A61K31/5377;A61K45/00;A61P1/02;A61P1/16;A61P9/10;A61P11/00;A61P17/00;A61P17/06;A61P19/06;A61P25/28;A61P27/02;A61P29/00;A61P29/02;A61P31/12;A61P35/00;A61P37/00;A61P37/08;A61P43/00;C07D211/26;C07D211/32;C07D211/58;C07D401/06;C07D401/10;C07D401/12;C07D401/14;C07D405/06;C07D405/10;C07D405/12;C07D405/14;C07D409/06;C07D409/14;C07D411/00;C07D411/06;C07D413/10;C07D413/12;C07D413/14;C07D417/06;C07D471/04;C07D487/04;C07D495/04;C07D513/04;(IPC1-7):C07D401/06;C07D211/16;C07D401/04;A61K31/435 主分类号 A61K31/451
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