发明名称 HETEROARYL SUBSTITUTED TETRAZOLE MODULATORS OF METABOTROPIC GLUTAMATE RECEPTOR-5
摘要 Tetrazole compounds substituted directly, or by a bridge, with a heteroaryl moiety containing N adjacent to the point of connection of the heteroaryl, are mGluR5 modulators useful in the treatment of psychiatric and mood disorders such as, for example, schizophrenia, anxiety, depression, and panic, as well as in the treatment of pain and other diseases.
申请公布号 WO03029210(A2) 申请公布日期 2003.04.10
申请号 WO2002US31294 申请日期 2002.10.01
申请人 MERCK & CO. INC.;COSFORD, NICHOLAS, D.;ROPPE, JEFFREY;CHEN, CHIXU;SMITH, NICHOLAS;REGER, THOMAS 发明人 COSFORD, NICHOLAS, D.;ROPPE, JEFFREY;CHEN, CHIXU;SMITH, NICHOLAS;REGER, THOMAS
分类号 A61K31/135;A61K31/4155;A61K31/4178;A61K31/4184;A61K31/42;A61K31/422;A61K31/4439;A61K31/4709;A61K31/4725;A61K31/485;A61K31/497;A61K45/00;A61P3/04;A61P25/04;A61P25/08;A61P25/14;A61P25/16;A61P25/18;A61P25/20;A61P25/22;A61P25/24;A61P25/28;A61P25/30;A61P25/34;A61P29/00;C07D401/04;C07D401/14;C07D403/04;C07D403/14;C07D405/04;C07D405/14;C07D413/04;C07D413/14;C07D417/04;C07D417/14;C07D471/04 主分类号 A61K31/135
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