发明名称 LOW HYGROSCOPIC ARIPIPRAZOLE DRUN SUBSTANCE AND PROCESSES FOR THE PREPARATION THEREOF
摘要 The present invention provides low-hygroscopic forms of aripiprazole and processes for the preparation thereof which will not convert to a hydrate or lose their original solubility even when a medicinal preparation containing the aripiprazole anhydride crystals is stored for an extended period.
申请公布号 CA2689052(A1) 申请公布日期 2003.04.03
申请号 CA20022689052 申请日期 2002.09.25
申请人 OTSUKA PHARMACEUTICAL CO., LTD. 发明人 ABE, KAORU;AOKI, SATOSHI;KAWASAKI, JUNICHI;TANIGUCHI, YOUICHI;BANDO, TAKUJI;TAKAHASHI, MASANORI;YABUUCHI, TSUYOSHI;ISHIGAMI, MAKOTO;NAKAGAWA, TOMONORI;SHINHAMA, KOICHI;FUJIMOTO, KIYOSHI;UTSUMI, NAOTO;OOI, YOSHIHIRO;FUJIMURA, TSUTOMU;NISHIOKA, YOSHIHIRO;KOBAYASHI, NORIYUKI;TOMIKAWA, KENJI;TOMINAGA, MICHIAKI;YAMADA, SHOHEI
分类号 C07D215/22;A61J3/02;A61K;A61K9/14;A61K9/16;A61K9/20;A61K31/4704;A61K31/496;A61K31/501;A61P;A61P1/08;A61P3/04;A61P15/10;A61P25/00;A61P25/04;A61P25/16;A61P25/18;A61P25/22;A61P25/28;A61P25/32;B01D9/02;C07D;C07D215/227;C07D401/12 主分类号 C07D215/22
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