发明名称 |
7-TERT-BUTYL-3-(2-FLUOROPHENYL)-6-(2H-(1,2,4)TRIAZOL-3-YLMETHOXY)-(1,2,4)TRIAZOLO (4,3-B) PYRIDAZINE FOR THE TREATMENT OF ANXIETY AND CONVULSIONS |
摘要 |
The compound (I) is a GABAa receptor ligand, functionally selective for the alpha 2 and/or alpha 3 subunit, and is useful in the treatment of deleterious mental states, in particular anxiety.
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申请公布号 |
WO03024968(A1) |
申请公布日期 |
2003.03.27 |
申请号 |
WO2002GB04201 |
申请日期 |
2002.09.13 |
申请人 |
MERCK SHARP & DOHME LIMITED;CARLING, WILLIAM, ROBERT;MOORE, KEVIN, WILLIAM;STREET, LESLIE, JOSEPH |
发明人 |
CARLING, WILLIAM, ROBERT;MOORE, KEVIN, WILLIAM;STREET, LESLIE, JOSEPH |
分类号 |
A61K31/519;A61P25/00;A61P25/08;A61P25/22;C07D487/04;(IPC1-7):C07D487/04;A61K31/502 |
主分类号 |
A61K31/519 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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