发明名称 THIOPHENYLTHIOPYRANE DIOXIDES AS MMP OR TNF-ALPHA INHIBITORS
摘要 A compound of the formula : in which R<1> is optionally substituted phenyl, optionally substituted naphthyl, optionally substituted bicyclic heterocyclic group, optionally substituted lower alkenyl or optionally substituted lower alkynyl, and R<2> is carboxy or protected carboxy, or a salt thereof, useful for treating and/or preventing MMP- or TNF- alpha mediated diseases.
申请公布号 WO03022842(A1) 申请公布日期 2003.03.20
申请号 WO2002JP08895 申请日期 2002.09.02
申请人 FUJISAWA PHARMACEUTICAL CO., LTD.;NEYA, MASAHIRO;SAWADA, AKIHIKO;OHNE, KAZUHIKO;ABE, YOSHITO;MIZUTANI, TSUYOSHI;ISHIBASHI, NAOKI;INOUE, MAKOTO 发明人 NEYA, MASAHIRO;SAWADA, AKIHIKO;OHNE, KAZUHIKO;ABE, YOSHITO;MIZUTANI, TSUYOSHI;ISHIBASHI, NAOKI;INOUE, MAKOTO
分类号 A61K31/382;A61K31/41;A61K31/4155;A61K31/422;A61K31/427;A61K31/4436;A61K31/4709;A61K31/497;A61P1/02;A61P9/10;A61P11/00;A61P17/00;A61P17/02;A61P17/06;A61P19/00;A61P19/02;A61P27/16;A61P29/00;A61P31/04;A61P31/18;A61P35/00;A61P37/08;A61P43/00;C07D409/04;C07D409/14;C07D413/14;C07D417/14;C07F7/08;C07F7/18;(IPC1-7):C07D409/04;A61K31/38 主分类号 A61K31/382
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