发明名称 METHOD FOR TREATING ALZHEIMER'S DISEASE USING QUINALDOYL-AMINE DERIVATIVES OF OXO- AND HYDROXY-SUBSTITUTED HYDROCARBONS
摘要 Disclosed are methods for treating Alzheimer's disease, and other diseases, and/or inhibiting beta-secretase enzyme, and/or inhibiting deposition of A beta peptide in a mammal, by use of compounds of formula (I), wherein R1, R2 , R3, and N* are defined herein.
申请公布号 CA2483959(A1) 申请公布日期 2003.03.13
申请号 CA20022483959 申请日期 2002.08.28
申请人 ELAN PHARMACEUTICALS, INC.;PHARMACIA & UPJOHN COMPANY LLC 发明人 SCHOSTAREZ, HEINRICH JOSEF
分类号 A61K45/00;A61K31/15;A61K31/165;A61K31/205;A61K31/27;A61K31/416;A61K31/4439;A61K31/47;A61K31/50;A61K31/502;A61K45/06;A61P25/00;A61P25/28;A61P43/00;(IPC1-7):A61K31/502;A61K31/440;A61K31/470;A61K31/501 主分类号 A61K45/00
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