发明名称 PENTAPEPTIDE COMPOUNDS AND USES RELATED THERETO
摘要 Pentapeptide compounds are disclosed. The compounds have biological activity, e.g. , cytotoxicity. Prodrugs having targeting groups and pentapeptide moieties, as well as precursors thereof are also disclosed. For example, precursors having a reactive linker that can serve as a reaction site for joining to a targeting agent, e.g. , an antibody, as disclosed.
申请公布号 WO02088172(A3) 申请公布日期 2003.02.27
申请号 WO2002US13435 申请日期 2002.04.30
申请人 SEATTLE GENETICS, INC.;DORONINA, SVETLANA;SENTER, PETER, D.;TOKI, BRIAN, E. 发明人 DORONINA, SVETLANA;SENTER, PETER, D.;TOKI, BRIAN, E.
分类号 A61K38/00;A61P35/00;A61P37/02;A61P43/00;C07K5/02;C07K5/03 主分类号 A61K38/00
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