发明名称 2H-PHTHALAZIN-1-ONES AND METHODS FOR USE THEREOF
摘要 The present invention provides compounds comprising a bicyclic aryl moiety, such as 2H-phthalazin-1-one or derivatives thereof, compositions comprising the same, and methods for producing and using the same. In particular, the present invention provides compounds of the formula: (I) or a pharmaceutically acceptable salt, a hydrate, a solvate, or a prodrug thereof; where Q<1>, Q<2> and Y are those defined herein.
申请公布号 WO03015785(A1) 申请公布日期 2003.02.27
申请号 WO2002US26271 申请日期 2002.08.15
申请人 ICOS CORPORATION;BEATON, GRAHAM;MOREE, WILNA, J.;RUETER, JAIMIE, K.;DAHL, RUSSELL, S.;MCELLIGOTT, DAVID, L.;GOLDMAN, PHYLLIS;DEMAGGIO, ANTHONY, J.;CHRISTENSON, ERIK;HERENDEEN, DAN;FOWLER, KERRY, W.;HUANG, DANWEN;BERTINO, JAIMIE, A.;BOURDON, LISA, H.;FAIRFAX, DAVID, J.;JIANG, QIN;REISCH, HELGE, A.;SONG, REN, HUA;ZHICHKIN, PAVEL, E. 发明人 BEATON, GRAHAM;MOREE, WILNA, J.;RUETER, JAIMIE, K.;DAHL, RUSSELL, S.;MCELLIGOTT, DAVID, L.;GOLDMAN, PHYLLIS;DEMAGGIO, ANTHONY, J.;CHRISTENSON, ERIK;HERENDEEN, DAN;FOWLER, KERRY, W.;HUANG, DANWEN;BERTINO, JAIMIE, A.;BOURDON, LISA, H.;FAIRFAX, DAVID, J.;JIANG, QIN;REISCH, HELGE, A.;SONG, REN, HUA;ZHICHKIN, PAVEL, E.
分类号 A61K31/502;A61K31/5025;A61K31/5377;A61K41/00;A61K49/00;A61P9/00;A61P9/10;A61P25/00;A61P25/14;A61P25/16;A61P25/28;A61P35/00;A61P43/00;C07D237/32;C07D237/34;C07D241/44;C07D401/12;C07D403/12;C07D405/12;C07D413/12;C07D413/14;C07D417/14;C07D471/04;C07D487/04;(IPC1-7):A61K31/502 主分类号 A61K31/502
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