发明名称 Aminoalcohol derivatives
摘要 A compound of the formula [Ig]; wherein R1 is hydrogen or an amino protective group, R2 is hydrogen or hydroxy, and R3 and R4 are independently N-methyl-methoxycarbonylamino, N-ethyl-methoxycarbonylamino, N-propyl-methoxycarbonylamino or 3-ethylureid, or R3 and R4 are both methoxycarbonylamino substituted at a meta position of the benzene rings, or a salt thereof, and (2S)-1-phenoxy-3-[3,3-bis[4-methoxycarbonylamino)-phenyl]propylamino]-2-propanol sulfate (2:1) and some crystal forms thereof as beta3adrenergic receptor agonists.
申请公布号 US2003032834(A1) 申请公布日期 2003.02.13
申请号 US20020203626 申请日期 2002.08.19
申请人 KAYAKIRI HIROSHI;FUJII NAOAKI;HAMASHIMA HITOSHI;SAKURAI MINORU;WASHIZUKA KENICHI;TOMISHIMA YASUYO;TANIGUCHI KIYOSHI;UNAMI NAOKO;KONO YUTAKA;ISHIKAWA HIROFUMI;YAMAMOTO NOBUHIRO;MIMURA HISASHI 发明人 KAYAKIRI HIROSHI;FUJII NAOAKI;HAMASHIMA HITOSHI;SAKURAI MINORU;WASHIZUKA KENICHI;TOMISHIMA YASUYO;TANIGUCHI KIYOSHI;UNAMI NAOKO;KONO YUTAKA;ISHIKAWA HIROFUMI;YAMAMOTO NOBUHIRO;MIMURA HISASHI
分类号 A61P1/04;A61K31/17;A61K31/27;A61P1/06;A61P1/16;A61P1/18;A61P3/04;A61P3/06;A61P3/10;A61P9/10;A61P9/12;A61P13/00;A61P13/04;A61P13/08;A61P13/10;A61P25/02;A61P25/24;A61P27/06;A61P43/00;C07C269/06;C07C271/28;(IPC1-7):C07C271/28;A61K31/325 主分类号 A61P1/04
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