发明名称 BENZOXAZOLE LPAAT- BETA INHIBITORS AND USES THEREOF
摘要 The invention relates to benzoxazoles of the following Formula, wherein the variables are defined in the claims and the use thereof to inhibit lysophosphatidic acid acyltransferase beta (LPAAT- beta ) activity. The invention further relates to methods of treating cancer using said benzoxazoles. The invention also relates to methods for screening to LPAAT- beta activitiy.
申请公布号 WO0236580(A9) 申请公布日期 2003.02.13
申请号 WO2001US42836 申请日期 2001.10.30
申请人 BONHAM, LYNN;LEUNG, DAVID, W.;HOLLENBACK, DAVID, M.;KLEIN, J., PETER;FINNEY, ROBERT, E.;WHITE, THAYER, H.;SHAFFER, SCOTT, A.;TANG, NORINA, M. 发明人 BONHAM, LYNN;LEUNG, DAVID, W.;HOLLENBACK, DAVID, M.;KLEIN, J., PETER;FINNEY, ROBERT, E.;WHITE, THAYER, H.;SHAFFER, SCOTT, A.;TANG, NORINA, M.
分类号 A61P35/00;C07D235/18;C07D263/56;C07D263/57;C07D277/66;(IPC1-7):C07D263/57;C07D498/04;C07D513/04;A61K31/423 主分类号 A61P35/00
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