发明名称 1,2,5,6-tetrahydro-4H-imidazo[4,5,1-ij]-quinolin-2(1H)-one derivatives
摘要 A tricyclic compound of formula (II), where: RN is selected from the group consisting of: (A) phenyl-CH2- where phenyl is optionally substituted with 1 or 2 of alkoxy, F, Cl, Br, I or alkyl; (B) RN1-CH2-O-CH2- where RN1 is selected from the group consisting of: phenyl which is optionally substituted with alkyl, F, Cl, Br, I or alkoxy; (CH3)3Si-CH2-; RN2-O-CH2- where RN2 is alkyl; CH2=CH-; H; or alkyl; (C) CH2=CH-CH2-, CH3-CH=CH-CH2-, or phenyl-CH=CH-CH2-. Also described is a hydroxy compound of formula (III) where RN has the same meaning as defined above and where RX is Br, Cl or I. Also described is an ester of formula (IV) where RN and RX have the same meanings as defined above. Also described is a hydroxy-amino compound of formula (V) where RN has the same meaning as defined above. Also described is tetracyclic compound of formula (VI), where RN has the same meaning as defined above.
申请公布号 NZ513347(A) 申请公布日期 2003.01.31
申请号 NZ20000513347 申请日期 2000.01.31
申请人 PHARMACIA & UPJOHN COMPANY 发明人 WUTS, PETER GUILLAUME MARIE
分类号 C07D471/06;C07D471/16;(IPC1-7):C07D471/06 主分类号 C07D471/06
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