发明名称 |
PREPARATION OF [1S-[1a, 2b, 3b, 4a(S*)]-4-[7[[ [1-(3-CHLOR-2-THIENYL)METHYL]PROPYL]AMINO]-3H-IMIDAZO[4,5-b]PYRIDIN -3-YL]-N-ETHYL-2,3-DIHYDROXYCYCLOPENTANE CARBOXAMIDE |
摘要 |
The invention relates to methods for the preparation of [1s-[1a, 2b, 3b, 4a(S*)]-4-[7- [[1-(3-chlor-2-thienyl)methyl]propyl]amino]-3H-imidazo[4,5-b]pyrid in-3-yl]-N-ethyl-2,3-dihydroxycyclopentane carboxamide, to methods for the preparation of its intermediate compounds and to the above intermediate compounds. 27 claims
|
申请公布号 |
BG63805(B1) |
申请公布日期 |
2003.01.31 |
申请号 |
BG19990103484 |
申请日期 |
1999.06.11 |
申请人 |
AVENTIS PHARMACEUTICALS INC |
发明人 |
O'BRIAN, MICHAEL K.;GARCIA, HERVE;LEON, PATRICK;POWNER, TORY H.;REILLY, LAURENCE W.;SHAH, HARSHAVADAN C.;THOMPSON, MICHAEL D.;TSUEI, CHING T.;VANASSE, BENOIT J.;WALTHER, FRANCIS L. |
分类号 |
A61P3/06;A61P9/00;A61P9/12;C07D213/69;C07D409/12;C07D409/14;C07D471/04;(IPC1-7):C07D471/04;C07D213/00;C07D213/62 |
主分类号 |
A61P3/06 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|