发明名称 PREPARATION OF [1S-[1a, 2b, 3b, 4a(S*)]-4-[7[[ [1-(3-CHLOR-2-THIENYL)METHYL]PROPYL]AMINO]-3H-IMIDAZO[4,5-b]PYRIDIN -3-YL]-N-ETHYL-2,3-DIHYDROXYCYCLOPENTANE CARBOXAMIDE
摘要 The invention relates to methods for the preparation of [1s-[1a, 2b, 3b, 4a(S*)]-4-[7- [[1-(3-chlor-2-thienyl)methyl]propyl]amino]-3H-imidazo[4,5-b]pyrid in-3-yl]-N-ethyl-2,3-dihydroxycyclopentane carboxamide, to methods for the preparation of its intermediate compounds and to the above intermediate compounds. 27 claims
申请公布号 BG63805(B1) 申请公布日期 2003.01.31
申请号 BG19990103484 申请日期 1999.06.11
申请人 AVENTIS PHARMACEUTICALS INC 发明人 O'BRIAN, MICHAEL K.;GARCIA, HERVE;LEON, PATRICK;POWNER, TORY H.;REILLY, LAURENCE W.;SHAH, HARSHAVADAN C.;THOMPSON, MICHAEL D.;TSUEI, CHING T.;VANASSE, BENOIT J.;WALTHER, FRANCIS L.
分类号 A61P3/06;A61P9/00;A61P9/12;C07D213/69;C07D409/12;C07D409/14;C07D471/04;(IPC1-7):C07D471/04;C07D213/00;C07D213/62 主分类号 A61P3/06
代理机构 代理人
主权项
地址