SELECTIVE ANDROGEN RECEPTOR MODULATORS AND METHODS FOR THEIR IDENTIFICATION, DESIGN AND USE
摘要
Selective androgen receptor modulators (SARMs) having antagonist activity in hormone-dependent tumors while exhibiting no activity or agonist activity against other nontumor tissues containing the androgen receptor as well as methods for identifying, designing and using SARMs are provided.
申请公布号
WO0200617(A3)
申请公布日期
2003.01.30
申请号
WO2001US19665
申请日期
2001.06.20
申请人
BRISTOL-MYERS SQUIBB COMPANY;SALVATI, MARK, E.;GOTTARDIS, MARCO, M.;KRYSTEK, STANLEY, R., JR.;ATTAR, RICARDO, M.;SACK, JOHN, S.
发明人
SALVATI, MARK, E.;GOTTARDIS, MARCO, M.;KRYSTEK, STANLEY, R., JR.;ATTAR, RICARDO, M.;SACK, JOHN, S.